Therapeutic Targeting of the Pyruvate Dehydrogenase ... | 食品添加物合法業者資訊網
由PWStacpoole著作·2017·被引用137次—Themitochondrialpyruvatedehydrogenasecomplex(PDC)irreversiblydecarboxylatespyruvatetoacetylcoenzymeA,therebylinkingglycolysis ...
The mitochondrial pyruvate dehydrogenase complex (PDC) irreversibly decarboxylates pyruvate to acetyl coenzyme A, thereby linking glycolysis to the tricarboxylic acid cycle and defining a critical step in cellular bioenergetics. Inhibition of PDC activity by pyruvate dehydrogenase kinase (PDK)-mediated phosphorylation has been associated with the pathobiology of many disorders of metabolic integration, including cancer. Consequently, the PDC/PDK axis has long been a therapeutic target. The most common underlying mechanism accounting for PDC inhibition in these conditions is post-transcriptional upregulation of one or more PDK isoforms, leading to phosphorylation of the E1α subunit of PDC. Such perturbations of the PDC/PDK axis induce a "glycolytic shift," whereby affected cells favor adenosine triphosphate production by glycolysis over mitochondrial oxidative phosphorylation and cellular proliferation over cellular ...
Distinct regulatory properties of pyruvate dehydrogenase ... | 食品添加物合法業者資訊網
Pyruvate Dehydrogenase Kinase | 食品添加物合法業者資訊網
Pyruvate dehydrogenase kinase | 食品添加物合法業者資訊網
Pyruvate dehydrogenase kinase as a novel ... | 食品添加物合法業者資訊網
Pyruvate Dehydrogenase Kinase Is a Metabolic ... | 食品添加物合法業者資訊網
Pyruvate dehydrogenase kinase regulatory mechanisms and ... | 食品添加物合法業者資訊網
The pivotal role of pyruvate dehydrogenase kinases in ... | 食品添加物合法業者資訊網
Therapeutic potential of the mammalian pyruvate ... | 食品添加物合法業者資訊網
Therapeutic Targeting of the Pyruvate Dehydrogenase ... | 食品添加物合法業者資訊網
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